Search results for "Multipolar spindles"

showing 3 items of 3 documents

Dis-organizing centrosomal clusters: specific cancer therapy for a generic spread?

2015

Cancer is a leading cause of mortality and the annual incidence of new cancer cases is rising worldwide. Due to the frequent development of resistance and the side effects of established anti-cancer drugs, the quest for new drugs with improved therapeutic features goes on. In contrast to cytotoxic chemotherapy of the past, the concept of targeted chemotherapy attempts to increase specificity of therapy by attacking tumor-related mechanisms. A novel emerging treatment concept represents the inhibition of centrosomal clustering. The centrosome regulates mitotic spindle formation assuring uniform separation of chromosomes to daughter cells. Many tumors contain supernumerary centrosomes, which …

PharmacologyCentrosomeBiological ProductsCell divisionColcemidOrganic ChemistryBiologyBiochemistrySpindle pole bodyVinblastineCell biologySpindle apparatusNocodazolechemistry.chemical_compoundchemistryCentrosomeNeoplasmsDrug DiscoverymedicineMolecular MedicineAnimalsHumansMultipolar spindlesmedicine.drugCurrent medicinal chemistry
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Centrosome structure is very similar in eupyrene and apyrene spermatocytes ofEphestia kuehniella(Pyralidae, Lepidoptera, Insecta)

1997

Summary The higher Lepidoptera produce two types of sperm, eupyrene and apyrene. Eupyrene spermatozoa are fertile, while apyrene spermatozoa are anucleate and, therefore, sterile. Meiosis differs between the two developmental lines. One of the most obvious differences is the aberrant organization of the apyrene spindles. They possess fewer microtubules than eupyrene spindles and chromosome segregation is irregular. To determine whether micotubule nucleation is impaired in the aprene spindles, the present fine structure study concentrated on the centrosomes in both spermatocyte types. In addition, the presence of gamma-tubulin, a newly discovered tubulin isoform which is prevalent in centros…

GeneticsbiologySpermatocyteCell biologyChromosome segregationmedicine.anatomical_structureTubulinMeiosisMicrotubuleCentrosomemedicinebiology.proteinAnimal Science and ZoologySpermatogenesisMultipolar spindlesDevelopmental BiologyInvertebrate Reproduction & Development
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A selective inhibitor of the Polo-box domain of Polo-like kinase 1 identified by virtual screening

2018

Graphical abstract

0301 basic medicineLK Polo-like kinasePolo-like kinaseCell cycleIC50 50% inhibition concentrationVirtual drug screeningPLK103 medical and health sciences0302 clinical medicineNeoplasmsTargeted chemotherapylcsh:Science (General)MitosisComputingMethodologies_COMPUTERGRAPHICSCDK cyclin-dependent kinasePBD Polo-box domainPyRxNatural productslcsh:R5-920MultidisciplinaryMicroscale thermophoresisKinaseChemistryCell cycleCell biology030104 developmental biology030220 oncology & carcinogenesisCancer cellOriginal ArticleCAMKK2 calcium/calmodulin-dependent protein kinase kinase 2PC Polo-box caplcsh:Medicine (General)Multipolar spindleslcsh:Q1-390Journal of Advanced Research
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